Xavier Dezitter
Publications
Article dans une revue scientifique
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Douguet, Laetitia
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Janho Dit Hreich, Serena
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Benzaquen, J.
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Seguin, L.
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Juhel, T.
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Dezitter, Xavier
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Duranton, C.
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Ryffel, B.
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Kanellopoulos, Jean
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Delarasse, Cecile
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Renault, Nicolas
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Furman, Christophe
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Homerin, Germain
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Féral, C.
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Cherfils-Vicini, J.
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Millet, Régis
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Adriouch, Sahil
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Ghinet, Alina
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Hofman, P.
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Vouret-Craviari, V.
A small-molecule P2RX7 activator promotes anti-tumor immune responses and sensitizes lung tumor to immunotherapy.
Nature Communications, 2021 , https://dx.doi.org/10.1038/s41467-021-20912-2
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Homerin, Germain
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Jawhara, Samir
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Dezitter, Xavier
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Baudelet, Davy
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Dufrénoy, Pierrick
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Rigo, Benoît
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MILLET, Régis
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Furman, Christophe
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Ragé, Guillaume
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Lipka, Emmanuelle
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Farce, Amaury
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Renault, Nicolas
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Sendid, Boualem
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Charlet, Rogatien
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Leroy, Jordan
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Phanithavong, Mélodie
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Richeval, Camille
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Wiart, Jean-François
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Allorge, Delphine
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Adriouch, Sahil
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Vouret-Craviari, Valérie
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Ghinet, Alina
Pyroglutamide-Based P2X7 Receptor Antagonists Targeting Inflammatory Bowel Disease
Journal of Medicinal Chemistry, American Chemical Society (ACS), 2019 , https://dx.doi.org/10.1021/acs.jmedchem.9b00584
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Sikkeland, Jorgen
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Lindstad, Torstein
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Nenseth, Hatice Zeynep
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Dezitter, Xavier
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Qu, Su
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Muhumed, Ridhwan M.
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Ertunc, Meric Erikci
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Gregor, Margaret F.
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Saatcioglu, Fahri
Inflammation and er stress differentially regulate stamp2 expression and localization in adipocytes
Metabolism. clinical and experimental, 2019 , https://dx.doi.org/10.1016/j.metabol.2019.01.014
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Sansook, Supojjanee
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Tuo, Wei
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Bollier, Melanie
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Barczyk, Amélie
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Dezitter, Xavier
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Klupsch, Frederique
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Chavain, Natascha
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Farce, Amaury
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Tizzard, Graham J.
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Coles, Simon J.
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Spencer, John
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Millet, Régis
Synthesis and biological evaluation of ferrocene-based cannabinoid receptor 2 ligands
Future Medicinal Chemistry, 2018 , https://dx.doi.org/10.4155/fmc-2017-0200
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Tuo, Wei
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Bollier, Melanie
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Chavain, Natascha
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Lemaire, Lucas
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Barczyk, Amélie
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Dezitter, Xavier
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Klupsch, Frederique
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Szczepanski, Fabien
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Spencer, John
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Chavatte, Philippe
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Millet, Régis
Development of novel oxazolo[5,4-d]pyrimidines as competitive cb2 neutral antagonists based on scaffold hopping
European Journal of Medicinal Chemistry, 2018 , https://dx.doi.org/10.1016/j.ejmech.2018.01.034
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Homerin, Germain
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Lipka, Emmanuelle
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Rigo, Benoit
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MILLET, Régis
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Dezitter, Xavier
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Furman, Christophe
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Ghinet, Alina
Discovery of highly functionalized scaffolds: Pyrroloimidazolediones as P2X7 receptor antagonists
Tetrahedron, 2017 , https://dx.doi.org/10.1016/j.tet.2017.07.036
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Tesikova, Martina
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Dezitter, Xavier
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Nenseth, Hatice Z.
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Klokk, Tove I.
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Mueller, Florian
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Hager, Gordon L.
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Saatcioglu, Fahri
Divergent Binding and Transactivation by Two Related Steroid Receptors at the Same Response Element
The Journal of biological chemistry, 2016 , https://dx.doi.org/10.1074/jbc.M115.684480
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Homerin, Germain
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Baudelet, Davy
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Dufrenoy, Pierrick
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Rigo, Benoit
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Lipka, Emmanuelle
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Dezitter, Xavier
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Furman, Christophe
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MILLET, Régis
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Ghinet, Alina
ZrCl4 as a new catalyst for ester amidation: an efficient synthesis of h-P2X7R antagonists
Tetrahedron Letters, 2016 , https://dx.doi.org/10.1016/j.tetlet.2016.02.004
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Baudelet, Davy
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Furman, Christophe
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Ghinet, Alina
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Dezitter, Xavier
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Adriouch, Sahil
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Capet, Frederic
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Rogez-Florent, Tiphaine
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Gautret, Philippe
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Rigo, Benoit
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Millet, Régis
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Vaccher, Claude
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Lipka, Emmanuelle
Evaluation and comparison of three different separation techniques for analysis of retroamide enantiomers and their biological evaluation against h-P2X7 receptor
Journal of chromatography. B, Analytical technologies in the biomedical and life sciences, 2015 , https://dx.doi.org/10.1016/j.jchromb.2015.02.001
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Baudelet, Davy
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Schifano, Nadege
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Ghinet, Alina
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Dezitter, Xavier
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Barbotin, Florent
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Gautret, Philippe
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Rigo, Benoit
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Chavatte, Philippe
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MILLET, Régis
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Furman, Christophe
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Vaccher, Claude
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Lipka, Emmanuelle
Enantioseparation of pyroglutamide derivatives on polysaccharide based chiral stationary phases by high-performance liquid chromatography and supercritical fluid chromatography: A comparative study
Journal of chromatography. A, 2014 , https://dx.doi.org/10.1016/j.chroma.2014.06.090
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Baudelet, Davy
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Ghinet, Alina
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Furman, Christophe
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Dezitter, Xavier
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Gautret, Philippe
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Rigo, Benoit
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MILLET, Régis
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Vaccher, Claude
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Lipka, Emmanuelle
Antagonists of the P2X7 receptor: Mechanism of enantioselective recognition using highly sulfated and sulfobutylether cyclodextrins by capillary electrokinetic chromatography
Electrophoresis, 2014 , https://dx.doi.org/10.1002/elps.201400113
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Nenseth, Hatice Z.
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Dezitter, Xavier
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Tesikova, Martina
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Mueller, Florian
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Klokk, Tove I.
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Hager, Gordon L.
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Saatcioglu, Fahri
Distinctly Different Dynamics and Kinetics of Two Steroid Receptors at the Same Response Elements in Living Cells
PLoS One, 2014 , https://dx.doi.org/10.1371/journal.pone.0105204
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Dezitter, Xavier
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Fagart, Jerome
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Taront, Solenne
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Fay, Michel
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Masselot, Bernadette
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Hetuin, Dominique
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Formstecher, Pierre
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Rafestin-Oblin, Marie-Edith
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Idziorek, Thierry
A Structural Explanation of the Effects of Dissociated Glucocorticoids on Glucocorticoid Receptor Transactivation
Molecular pharmacology, 2014 , https://dx.doi.org/10.1124/mol.113.085860
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Nhili, Raja
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Peixoto, Paul
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Depauw, Sabine
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Flajollet, Sebastien
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Dezitter, Xavier
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Munde, Manoj M.
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Ismail Mohamed, A.
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Kumar, Arvind
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Faraha, Abdelbasset A.
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Stephens, Chad E.
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Duterque-Coquillaud, Martine
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Wilson W., David
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Boykin, David W.
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David-Cordonnier, Marie-Helene
Targeting the DNA-binding activity of the human ERG transcription factor using new heterocyclic dithiophene diamidines
Nucleic acids research, 2013 , https://dx.doi.org/10.1093/nar/gks971
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Joha, S
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Nugues, A-L
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Hetuin, D
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Berthon, Celine
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Dezitter, Xavier
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Dauphin, V
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Mahon, F-X
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Roche-Lestienne, C
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Preudhomme, Claude
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Quesnel, Bruno
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Idziorek, Thierry
GILZ inhibits the mTORC2/AKT pathway in BCR-ABL(+) cells
Oncogene, 2012 , https://dx.doi.org/10.1038/onc.2011.328
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Dezitter, Xavier
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Masselot, Bernadette
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Tardivel, Meryem
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Mereau-Richard, Claude
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Formstecher, Pierre
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Idziorek, Thierry
Macromolecular synthesis inhibitors perturb glucocorticoid receptor trafficking
The Journal of steroid biochemistry and molecular biology, 2011 , https://dx.doi.org/10.1016/j.jsbmb.2011.04.008
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Dezitter, Xavier
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Hammoudi, Fatma
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Belverge, Nicolas
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Deloulme, Jean-Christophe
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Drobecq, Herve
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Masselot, Bernadette
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Formstecher, Pierre
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Mendy, Denise
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Idziorek, Thierry
Proteomics unveil corticoid-induced S100A11 shuttling in keratinocyte differentiation
Biochemical and biophysical research communications, 2007 , https://dx.doi.org/10.1016/j.bbrc.2007.06.113
Brevet
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Vouret-Craviari, Valerie
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Douguet, Laetitia
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Ghinet, Alina
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Homerin, Germain
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Rigo, Benoît
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Baudelet, Davy
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Dezitter, Xavier
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Millet, Régis
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Furman, Christophe
P2rx7 modulators in therapy
WO2019185868A1, France, 2019,
Compte-rendu et recension critique d'ouvrage
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Le Biannic, Raphaël
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Magnez, Romain
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Klupsch, Frédérique
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Leleu-Chavain, Natascha
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Thiroux, Bryan
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Tardy, Morgane
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El Bouazzati, Hassiba
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Dezitter, Xavier
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Renault, Nicolas
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Vergoten, Gérard
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Bailly, Christian
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Quesnel, Bruno
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Thuru, Xavier
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Millet, Régis
Pyrazolones as inhibitors of immune checkpoint blocking the PD-1/PD-L1 interaction
Elsevier, 2022, , https://dx.doi.org/10.1016/j.ejmech.2022.114343
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Le Biannic, Raphaël
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Magnez, Romain
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Klupsch, Frédérique
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Leleu-Chavain, Natascha
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Thiroux, Bryan
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Tardy, Morgane
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El Bouazzati, Hassiba
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Dezitter, Xavier
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Renault, Nicolas
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Vergoten, Gérard
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Bailly, Christian
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Quesnel, Bruno
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Thuru, Xavier
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Millet, Régis
Pyrazolones as inhibitors of immune checkpoint blocking the PD-1/PD-L1 interaction
Elsevier, 2022, , https://dx.doi.org/10.1016/j.ejmech.2022.114343