nicolas Willand
Publications
Compte-rendu et recension critique d'ouvrage
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Tatum, Natalie
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Villemagne, Baptiste
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Willand, nicolas
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Deprez, Benoit
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Liebeschuetz, John
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Baulard, Alain
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Pohl, Ehmke
Structural and docking studies of potent ethionamide boosters
International Union of Crystallography, 2013, , https://dx.doi.org/10.1107/S0108270113028126
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Flipo, Marion
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Willand, nicolas
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Lecat-Guillet, Nathalie
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Hounsou, Candide
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Desroses, Matthieu
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Leroux, Florence
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Lens, Zoé
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Villeret, Vincent
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Wohlkönig, Alexandre
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Wintjens, René
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Christophe, Thierry
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Kyoung Jeon, Hee
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Locht, Camille
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Brodin, Priscille
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Baulard, Alain
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Déprez, Benoit
Discovery of Novel N -Phenylphenoxyacetamide Derivatives as EthR Inhibitors and Ethionamide Boosters by Combining High-Throughput Screening and Synthesis
American Chemical Society, 2012, , https://dx.doi.org/10.1021/jm300377g
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Carette, Xavier
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Blondiaux, Nicolas
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Willery, Eve
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Hoos, Sylviane
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Lecat-Guillet, Nathalie
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Lens, Zoé
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Wohlkönig, Alexandre
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Wintjens, René
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Soror, Sameh
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Frénois, Frédéric
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Dirié, Bertrand
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Villeret, Vincent
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England, Patrick
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Lippens, Guy
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Deprez, Benoit
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Locht, Camille
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Willand, nicolas
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Baulard, Alain
Structural activation of the transcriptional repressor EthR from Mycobacterium tuberculosis by single amino acid change mimicking natural and synthetic ligands
Oxford University Press, 2011, , https://dx.doi.org/10.1093/nar/gkr1113
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Flipo, Marion
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Desroses, Matthieu
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Lecat-Guillet, Nathalie
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Villemagne, Baptiste
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Blondiaux, Nicolas
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Leroux, Florence
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Piveteau, Catherine
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Mathys, Vanessa
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Flament, Marie-Pierre
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Siepmann, Juergen
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Villeret, Vincent
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Wohlkönig, Alexandre
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Wintjens, René
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Soror, Sameh
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Christophe, Thierry
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Jeon, Hee Kyoung
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Locht, Camille
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Brodin, Priscille
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Déprez, Benoit
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Baulard, Alain
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Willand, nicolas
Ethionamide Boosters. 2. Combining Bioisosteric Replacement and Structure-Based Drug Design To Solve Pharmacokinetic Issues in a Series of Potent 1,2,4-Oxadiazole EthR Inhibitors
American Chemical Society, 2011, , https://dx.doi.org/10.1021/jm200825u
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Bonnel, David
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Legouffe, Raphael
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Willand, nicolas
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Baulard, Alain
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Hamm, Gregory
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Deprez, Benoit
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Stauber, Jonathan
MALDI imaging techniques dedicated to drug-distribution studies
Future Science, 2011, , https://dx.doi.org/10.4155/bio.11.88
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Flipo, Marion
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Desroses, Matthieu
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Lecat-Guillet, Nathalie
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Dirié, Bertrand
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Carette, Xavier
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Leroux, Florence
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Piveteau, Catherine
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Demirkaya, Fatma
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Lens, Zoé
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Rucktooa, Prakash
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Villeret, Vincent
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Christophe, Thierry
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Jeon, Hee Kyoung
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Locht, Camille
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Brodin, Priscille
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Déprez, Benoit
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Baulard, Alain
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Willand, nicolas
Ethionamide Boosters: Synthesis, Biological Activity, and Structure−Activity Relationships of a Series of 1,2,4-Oxadiazole EthR Inhibitors
American Chemical Society, 2011, , https://dx.doi.org/10.1021/jm200076a
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Willand, nicolas
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Desroses, Matthieu
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Toto, Patrick
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Dirié, Bertrand
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Lens, Zoé
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Villeret, Vincent
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Rucktooa, Prakash
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Locht, Camille
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Baulard, Alain
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Deprez, Benoit
Exploring Drug Target Flexibility Using in Situ Click Chemistry: Application to a Mycobacterial Transcriptional Regulator
American Chemical Society, 2010, , https://dx.doi.org/10.1021/cb100177g
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Willand, nicolas
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Dirié, Bertrand
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Carette, Xavier
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Bifani, Pablo
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Singhal, Amit
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Desroses, Matthieu
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Leroux, Florence
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Willery, Eve
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Mathys, Vanessa
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Déprez-Poulain, Rebecca
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Delcroix, Guy
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Frénois, Frédéric
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Aumercier, Marc
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Locht, Camille
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Villeret, Vincent
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Déprez, Benoit
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Baulard, Alain
Synthetic EthR inhibitors boost antituberculous activity of ethionamide
Nature Publishing Group, 2009, , https://dx.doi.org/10.1038/nm.1950
Partie d'ouvrage
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Willand, nicolas
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Flipo, Marion
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Villemagne, Baptiste
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Baulard, Alain
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Deprez, Benoit
Recent advances in the design of inhibitors of mycobacterial transcriptional regulators to boost thioamides anti-tubercular activity and circumvent acquired-resistance
Medicinal Chemistry Approaches to Tuberculosis and Trypanosomiasis, 2019, , https://dx.doi.org/10.1016/bs.armc.2019.06.003